Table 1.
Summary of in vitro data from first focused library.
![]() | ||
|---|---|---|
| Compound | R | IC50 (μM) |
| 1 | ![]() |
0.105 |
| 2 | ![]() |
0.11 |
| 7a | ![]() |
0.31 |
| 7b | ![]() |
0.97 |
| 7c | ![]() |
1.22 |
| 7d | ![]() |
1.83 |
| 7e | ![]() |
1.96 |
| 7f | ![]() |
3.55 |
| 7g | ![]() |
4.28 |
| 7h | ![]() |
4.90 |
| 7i | ![]() |
5.00 |
| 7j | ![]() |
10.69 |
| 7k | ![]() |
11.92 |
| 7l | ![]() |
26.18 |
| 7m | ![]() |
45.49 |
| 7n | ![]() |
>100 |
| 70 | ![]() |
>100 |
| 7p | ![]() |
>100 |


















