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. Author manuscript; available in PMC: 2010 Apr 2.
Published in final edited form as: Org Lett. 2009 Apr 2;11(7):1651–1654. doi: 10.1021/ol900306v

Table 2.

Dehydrogenative Coupling of Indolesa

graphic file with name nihms-103280-t0003.jpg

entry indole R1 R2 R3 yield (%)b
1 9a H H H 81
2 9b 5-OMe H H 86
3 9c 5-Br H H 76
4 9d 5-CO2Me H H 73
5 9e 4-Br H H 74
6 9f H H CO2Me 70
7 9g H H Me 63
8 9h 7-Me H H 0
9 9i H Me H 0
a

See Supporting Information for full experimental details.

b

Isolated yield.