Table 2.
entry | indole | R1 | R2 | R3 | yield (%)b |
---|---|---|---|---|---|
1 | 9a | H | H | H | 81 |
2 | 9b | 5-OMe | H | H | 86 |
3 | 9c | 5-Br | H | H | 76 |
4 | 9d | 5-CO2Me | H | H | 73 |
5 | 9e | 4-Br | H | H | 74 |
6 | 9f | H | H | CO2Me | 70 |
7 | 9g | H | H | Me | 63 |
8 | 9h | 7-Me | H | H | 0 |
9 | 9i | H | Me | H | 0 |
See Supporting Information for full experimental details.
Isolated yield.