. Author manuscript; available in PMC: 2010 Nov 30.

Published in final edited form as: Respir Physiol Neurobiol. 2009 Aug 3;169(2):102–114. doi: 10.1016/j.resp.2009.07.014

TABLE 2.

Representative Adenosine Receptor Agonists and Antagonists

	A₁ Receptor	A_2A Receptor	A_2B Receptor	A₃ Receptor	Reference
Agonists	CHA, CCPA, S-ENBA, CVT-510	CGS-21680, HE-NECA, CVT-3146	NECA (non selective)	IB-MECA, 2-Cl-IB-MECA, DBXRM, VT160	Burnstock, 2007
Antagonists	DPCPX, N-0840, MRS1754, N-0840, WRC-0571	DMPX, KF17837, SCH58261, ZM241385, KW 6002	Enprofylline, MRE2029, F20, MRS17541, MRS 1706, 8-SPT, CGS15493, CVT-5440, IDPX	MRS1220, L-268605, MRS1191, MRS1523, VUF8504	Feoktisyov et al., 2001, Zablocki et al., 2005; Burnstock, 2007;

CCPA= chlorocyclopentyladenosine, CPA= cyclopentyladenosine, NECA= 5′-N-ethylcarboxyamido adenosine, CHA=cyclohexlyadenosine,