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. Author manuscript; available in PMC: 2009 Dec 4.
Published in final edited form as: Dev Neurobiol. 2008 May;68(6):729–743. doi: 10.1002/dneu.20615

Table 1.

Partial list of PET radiotracers

Target system or process Radiotracer
Neuroreceptor Systems
Dopaminergic Pre-synaptic dopamine pool 18F-fluoro-L-dopa, 18F-fluoro-L-m-tyrosine
D2 Dopamine receptors 11C-N-methylspiperone, 11C-raclopride
18F-spiperone, 18F-N-methylspiperone
D1 Dopamine receptors 11C-SCH23390
Dopamine reuptake sites 11C-nomifensine, 11C-cocaine, 18F-GBR
11C-carfentanil, 11C-diprenorphine
Opiate 18F-cyclofoxy
Benzodiazepine 11C-flumazenil
Serotonergic Pre-synaptic serotonin pool 11C-α-methyl-tryptophan
5-HT1A receptors 11C-WAY100,635
5-HT2A receptors 11C-MDL100,907, 18F-altanserin, 18F- setoperone
5-HT reuptake sites 11C-McN5652
MAO-B enzyme 11C-deprenyl
Amino acid transport, protein synthesis
11C-methionine, 11C-leucine, 11C-tyrosine
Tissue pH 11CO2, 11C-DMO
Tissue drug kinetics 11C-phenytoin, 11C-valproate, 13N-BCNU