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. Author manuscript; available in PMC: 2009 Dec 4.
Published in final edited form as: J Med Chem. 2008 Jul 17;51(15):4553–4562. doi: 10.1021/jm8001668

Figure 6.

Figure 6

Assessment of interaction of inhibitors with DNA by EtBr replacement assay. There is no binding of 25, 82, 67, and 189 at 100 μM with DNA (A). In contrast, EtBr is displaced from DNA by 192 in a concentration (0, 50, 100 μM) dependent manner (B).

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