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. Author manuscript; available in PMC: 2010 Dec 1.
Published in final edited form as: Toxicol Appl Pharmacol. 2009 Aug 19;241(2):135–142. doi: 10.1016/j.taap.2009.08.014

Table 3.

Parameters Utilized In the Coincubation Kinetic Model

Parameter Value Source
KDBTC 107,013 nM (k2BTC*Km)/(Vmax/[E]T)
(adapted from Masson et al., 2008)
k1BTC 0.65 nM−1min−1 optimization
k−1BTC 69,558 min−1 KDBTC*k1BTC
k2BTC 1,965 min−1 (Vmax/[E]T)/(1-(Vmax/[E]T)/k3BTC)
(adapted from Masson et al., 2008)
k3BTC 28,020 min−1 Stojan et al, 2002
KMBTC 100,000 nM Table 1
KDCPO 2.02 nM Table 2
k1CPO 0.7 nM−1min−1 optimization
k−1CPO 1.41 min−1 KDCPO*k1CPO
k2CPO 103 min−1 Table 2