. Author manuscript; available in PMC: 2010 Nov 12.

Published in final edited form as: J Med Chem. 2009 Nov 12;52(21):6716–6723. doi: 10.1021/jm901016k

Table 1.

21 most potent VHR screening hits (Ki value <20 μM).

#	Mol. Weight	Ki, μM
1	355.441	0.809
2	451.4374	1.76
3	332.3482	1.86
4	395.4902	2.01
5	261.338	2.09
6	364.1547	2.64
7	368.4522	2.94
8	268.2684	3.07
9	429.9075	3.13
10	377.2549	3.19
11	331.7759	3.49
12	442.8605	3.87
13	454.2384	4.44
14	395.2022	12.1
15	231.2506	12.8
16	385.0484	13.4
17	267.2404	13.8
18	352.3056	13.8
19	288.3204	15.8
20	359.208	15.9
21	481.2585	16.2

Compounds 11, 13, 19, and 21 are mixtures of E/Z-isomers.