TABLE 3.
Compd. | % inhibition at various concentrations in μg/ml | ||||||
---|---|---|---|---|---|---|---|
1000 | 500 | 250 | 100 | 50 | 25 | 10 | |
4a | 62.0 | 54.3 | 46.7 | 39.6 | 27.6 | 19.0 | 13.2 |
4b | 73.1 | 64.5 | 52.2 | 41.3 | 32.3 | 26.7 | 10.2 |
4c | 56.8 | 49.3 | 38.8 | 29.4 | 20.1 | 14.6 | 08.5 |
4d | 49.4 | 40.2 | 32.1 | 25.7 | 19.7 | 12.4 | 06.3 |
4e | 52.5 | 46.8 | 37.3 | 28.9 | 21.2 | 16.7 | 10.7 |
4f | 68.9 | 57.8 | 43.2 | 37.6 | 29.7 | 15.1 | 09.2 |
4g | 50.1 | 44.8 | 38.9 | 33.4 | 24.3 | 17.2 | 09.3 |
4h | 79.6 | 67.5 | 60.9 | 53.5 | 34.6 | 24.3 | 17.6 |
4i | 63.2 | 56.7 | 49.8 | 40.7 | 29.5 | 18.3 | 11.3 |
4j | 50.6 | 44.8 | 39.9 | 30.3 | 22.8 | 17.5 | 10.3 |
5a | 64.3 | 57.2 | 47.8 | 36.5 | 29.5 | 19.3 | 13.2 |
5b | 80.6 | 67.5 | 61.9 | 53.5 | 34.6 | 26.3 | 17.8 |
5c | 55.6 | 44.5 | 37.3 | 25.7 | 18.6 | 14.2 | 10.6 |
5d | 48.9 | 37.8 | 29.5 | 20.7 | 13.6 | 10.8 | 05.5 |
5e | 43.2 | 33.5 | 27.4 | 21.1 | 17.3 | 11.4 | 06.4 |
5f | 58.3 | 45.9 | 36.8 | 28.9 | 20.7 | 16.8 | 11.1 |
5g | 62.3 | 56.7 | 45.3 | 36.7 | 24.8 | 16.3 | 11.3 |
5h | 73.7 | 66.8 | 54.5 | 43.3 | 30.2 | 27.8 | 19.7 |
5I | 54.1 | 46.3 | 39.4 | 27.9 | 19.8 | 13.7 | 08.4 |
5j | 51.5 | 46.8 | 35.3 | 27.9 | 20.2 | 17.7 | 11.7 |
6a | 39.8 | 33.7 | 26.8 | 20.1 | 14.3 | 09.8 | 05.3 |
6b | 54.3 | 42.5 | 36.7 | 25.2 | 16.6 | 12.2 | 09.6 |
6c | 62.8 | 55.4 | 42.6 | 37.7 | 29.8 | 21.3 | 12.1 |
6d | 51.7 | 46.9 | 36.8 | 29.9 | 21.1 | 16.9 | 10.2 |
6e | 79.8 | 47.9 | 38.7 | 28.9 | 22.3 | 16.8 | 11.7 |
6f | 50.7 | 41.3 | 32.8 | 23.2 | 18.7 | 11.4 | 07.3 |
6g | 53.5 | 46.6 | 34.3 | 26.9 | 21.2 | 16.8 | 11.7 |
6h | 78.9 | 46.8 | 39.8 | 27.7 | 19.6 | 11.8 | 07.5 |
6i | 41.2 | 34.5 | 27.6 | 20.5 | 15.3 | 10.2 | 05.1 |
6j | 55.9 | 43.7 | 36.3 | 28.5 | 21.1 | 14.3 | 06.3 |