Table 4.
Compound | Aqueous Solubility (µM) |
---|---|
9e | 112 |
9l | 66 |
10h | 259 |
10i | 257 |
10j | 94 |
1 | 350 |
The relative aqueous solubilities were measured using a protocol based on Millipore’s MultiScreen aqueous solubility filter plate assay. Maximal solubility in this assay is 500 µM.