Table 2.
Peptide | kona | koff | KD | Apo-helicityb | Maximum helicityc |
---|---|---|---|---|---|
M−1 s−1 | s−1 | nM | % | % | |
VEK-30 | 4.54×105 | 2.93×10−2 | 65 | 34 | 74 |
VEK-30[D7A] | 1.26×105 | 5.61×10−2 | 446 | 29 | 58 |
VEK-30[D7N] | 3.62×104 | 7.04×10−2 | 1940 | 18 | 23 |
VEK-30[D7N/E9Q] | 5.04×104 | 8.60×10−2 | 1710 | 12 | 26 |
VEK-30[D7A/E9A] | 2.61×105 | 9.67×10−2 | 371 | 19 | 52 |
The association rate constant (kon) and dissociation rate constant (koff) were obtained by SPR and apparent equilibrium dissociation constants (KD) were calculated from the ratio of koff/kon.
% α-helix in absence of K2Pg.
% maximal attainable a-helix after titration with K2Pg.