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. 2010 Apr;77(4):678–686. doi: 10.1124/mol.109.063065

TABLE 1.

NECA potency (Log EC50) in the absence and presence of antagonists and/or Brilliant Black BN at the adenosine A1 and A3 receptors

Data represent the mean ± S.E.M. of 3 to 11 experiments conducted in triplicate.

Brilliant Black BN
0 μM 5 μM 50 μM 500 μM
A1-CHO
    NECA −8.0 ± 0.3 −8.3 ± 0.3 −8.2 ± 0.2 −8.0 ± 0.1
    + 1 μM XAC-X-BY630 −7.3 ± 0.3 −7.7 ± 0.2 −7.9 ± 0.1 −8.0 ± 0.1
    + 1 μM XAC −7.0 ± 0.2 −7.3 ± 0.3 −7.7 ± 0.4 −7.9 ± 0.1
A3-CHO
    NECA −7.8 ± 0.2 −7.7 ± 0.2 −8.0 ± 0.2 −7.7 ± 0.1
    + 1 μM XAC-X-BY630 −6.7 ± 0.2 −6.5 ± 0.3 −7.2 ± 0.2 −7.5 ± 0.1
    + 1 μM XAC −6.7 ± 0.3 −6.4 ± 0.3 −7.4 ± 0.1 −7.4 ± 0.2