Figure 2.
Representative binding curves for Analogues Gal-B2 (triangles) and [N-Me, des-Sar]Gal-B2 (circles) against hGalR1 (left) and hGalR2 (right). Each binding assay was performed in triplicate to generate one 10-point binding curve. Binding affinities are reported as the average of three independent binding curves. Binding affinities (KI) for Gal-B2 are 3.5 nM hGalR1 and 52 nM hGalR2 and for [N-Me, des-Sar]Gal-B2 are 364 nM hGalR1 and 20 nM hGalR2.