Table 6.
In vitro inhibition of Notch cleavage by AD28 and AD115.
| Cpd | Conc. | In vitro Inhibition of Notch Cleavage |
|---|---|---|
| DMSO | 0.10% | - |
| DAPT | 100 μM | + |
| Gleevec | 100 μM | - |
| AD28 | 100 μM | + |
| AD94 | 100 μM | - |
| AD95 | 100 μM | - |
| AD115 | 100 μM | + |
In vitro inhibition of Notch cleavage by AD28 and AD115.
| Cpd | Conc. | In vitro Inhibition of Notch Cleavage |
|---|---|---|
| DMSO | 0.10% | - |
| DAPT | 100 μM | + |
| Gleevec | 100 μM | - |
| AD28 | 100 μM | + |
| AD94 | 100 μM | - |
| AD95 | 100 μM | - |
| AD115 | 100 μM | + |