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SAR study of narciclasine derivatives
| concen- tration |
[14C]Phe incorpo- ration |
concen- tration |
[3H]nar- ciclasine binding |
|
|---|---|---|---|---|
| compound | mM | % control | mM | % control |
| 44 | 0.1 | 6 | N/A | N/A |
| 1 | 0 | |||
| 49 | 0.1 | 8 | 0.01 | 25 |
| 1 | 5 | 1 | 4 | |
| 79 | 0.1 | 8 | 0.01 | 44 |
| 1 | 6 | 1 | 5 | |
| 77 | 0.1 | 67 | 0.1 | 96 |
| 1 | 52 | 1 | 90 | |
| 73 | 0.1 | 49 | 0.1 | 95 |
| 1 | 43 | 1 | 70 | |
| 78 | 0.1 | 21 | 0.1 | 68 |
| 1 | 12 | 1 | 16 | |
