TABLE 2.
Effect of adding radiolabeled precursors early on in vitro drug sensitivity tests
Time (h) of contact | Time (h) of freezing | Geometric mean IC50 in nM (95% CI)a |
|||
---|---|---|---|---|---|
T3/SAR97276 |
AS |
||||
HX | Ethanolamine | HX | Ethanolamine | ||
0-48 | 48 | 285.5 (151.9-536.9) | 38.5 (14.3-103.5) | 1.7 (1.3-2.2) | 1.7 (1.2-2.4) |
24-48 | 48 | 23.1 (15.5-34.4) | 22.3 (12.8-38.7) | 1.3 (1.2-1.5) | 0.9 (0.2-6) |
48-66 | 66 | 4.6 (4-5.2) | 9.4 (8.7-10.3) | 1.1 (0.8-1.4) | 1.5 (1.4-1.7) |
HX, hypoxanthine.