TABLE 1.
Polymerase and RT | IC50 (nM)a |
|||
---|---|---|---|---|
ETR | DAP | EFV | NVP | |
DDDP | ||||
WT | 126 ± 28 | 131 ± 23 | 57 ± 7 | 3.2 × 103 ± 4 × 102 |
M230L | 1,320 ± 31 | 1,290 ± 32 | 910 ± 26 | 156 × 103 ± 8 × 102 |
Fold change | 10.5 | 9.9 | 16 | 48.8 |
RDDP | ||||
WT | 68 ± 9 | 19 ± 3 | 30 ± 6 | 4.1 × 103 ± 3 × 102 |
M230L | 696 ± 27 | 172 ± 31 | 740 ± 35 | 185 × 103 ± 13 × 103 |
Fold change | 10.2 | 9.1 | 24.7 | 45.1 |
Data represent the means ± standard deviations of three separate determinations.