TABLE 1.
Na/K-ATPase inhibitors identified by high-throughput screen
These inhibitors produced at least 25% inhibition of Na/K-ATPase at 10 μg/ml.
Sample | Name | Formula |
---|---|---|
2006BD3 | Metacycline hydrochloride | C22H22N2O8.HCl |
2008BB8 | Tyrothricin | Mixture |
2018BF7 | Myricetin | C15H10O8 |
2021BG2 | Domiphen bromide | C22H40NO.Br |
2035BD1 | Resibufogenin | C24H32O4 |
2035BA5 | Cinobufagin | C26H34O6 |
2036BF1 | Oligomycin | C45H74O11 |
MB1 | 1,3-Dihydroxyxanthone | C13H8O4 |
MB2 | 3,4-Dihydroxyxanthone | C13H8O4 |
MB3 | 1,3,5-Trihydroxyxanthone | C13H8O5 |
MB5 | 3,4,5-Trihydroxyxanthone | C13H8O5 |
MB6 | 1,3,5,6-Tetrahydroxyxanthone | C13H8O6 |
MB7 | 3,4,5,6-Tetrahydroxyxanthone | C13H8O6 |