Skip to main content
. Author manuscript; available in PMC: 2011 Jun 7.
Published in final edited form as: Mol Pharm. 2010 Jun 7;7(3):689–698. doi: 10.1021/mp900259w

Table 1.

Rates and rates relative to vehicle (RRV) of EGFP-hAR transport for 4 doses of TEST, ANE, DHT, EPI, MET, NAN, OXA, and FLU and for VEH. Rate is min−1.

1 nM 10 nM 50 nM 100 nM
rate RRV rate RRV rate RRV rate RRV
TEST 0.0069 2.13 0.0134* 4.12 0.0525* 16.11 0.0301* 9.24
ANE 0.0029 0.90 0.0058 1.78 0.0157* 4.83 0.0112* 3.45
DHT 0.0012 0.38 0.0179* 5.51 0.0100* 3.06 0.0200* 6.15
EPI 0.0046 1.42 0.0096 2.96 0.0118* 3.63 0.0130* 4.00
MET 0.0114 3.50 0.0157* 4.81 0.0339* 10.41 0.0212* 6.51
NAN 0.0130* 4.00 0.0261* 8.03 0.0220* 6.76 0.0261* 8.01
OXA 0.0047 1.43 0.0213* 6.53 0.0276* 8.48 0.0196* 6.02
FLU 0.0059 1.80 0.0035 1.06 0.0153* 4.71 0.0033 1.02
VEH 0.0033 1.00
*

Rates significantly different from vehicle, p < 0.05.