Skip to main content
. 2009 Nov;158(Suppl 1):S44. doi: 10.1111/j.1476-5381.2009.00501_24.x
Nomenclature FFA1 FFA2 FFA3
Other names GPR40 (Sawzdargo et al., 1997) GPR43 (Sawzdargo et al., 1997) GPR41 (Sawzdargo et al., 1997) LSSIG (Senga et al., 2003)
Ensembl ID ENSG00000126266 ENSG00000126262 ENSG00000185897
Principal transduction Gq/11 (Briscoe et al., 2003; Itoh et al., 2003; Stoddart et al., 2007) Gq/11, Gi/o (Brown et al., 2003; Le Poul et al., 2003; Nilsson et al., 2003) Gi/o (Brown et al., 2003; Le Poul et al., 2003; Stoddart et al., 2007)
Selective agonists Linoleic acid (Briscoe et al., 2003); Itoh et al., 2003), GW9508 (pEC50 7.3; Briscoe et al., 2006; Sum et al., 2007), Cpd B (pEC50 6.1; Tan et al., 2008) (S)-2-(4-chlorophenyl)-N-(5-fluorothiazol-2-yl)-3-methylbutanamide (pEC50 6.4; Lee et al., 2008)
Selective antagonists GW1100 (Briscoe et al., 2006; Stoddart et al., 2007)