| Nomenclature | FFA1 | FFA2 | FFA3 |
| Other names | GPR40 (Sawzdargo et al., 1997) | GPR43 (Sawzdargo et al., 1997) | GPR41 (Sawzdargo et al., 1997) LSSIG (Senga et al., 2003) |
| Ensembl ID | ENSG00000126266 | ENSG00000126262 | ENSG00000185897 |
| Principal transduction | Gq/11 (Briscoe et al., 2003; Itoh et al., 2003; Stoddart et al., 2007) | Gq/11, Gi/o (Brown et al., 2003; Le Poul et al., 2003; Nilsson et al., 2003) | Gi/o (Brown et al., 2003; Le Poul et al., 2003; Stoddart et al., 2007) |
| Selective agonists | Linoleic acid (Briscoe et al., 2003); Itoh et al., 2003), GW9508 (pEC50 7.3; Briscoe et al., 2006; Sum et al., 2007), Cpd B (pEC50 6.1; Tan et al., 2008) | (S)-2-(4-chlorophenyl)-N-(5-fluorothiazol-2-yl)-3-methylbutanamide (pEC50 6.4; Lee et al., 2008) | – |
| Selective antagonists | GW1100 (Briscoe et al., 2006; Stoddart et al., 2007) | – | – |