Table 5.
Phase II combination studies of bortezomib
Patient population | Metastatic colorectal cancer | Metastatic pancreatic carcinoma | Pretreated NSCLC |
---|---|---|---|
Number of patients | 68 | 87 | 155 |
Schedule | Arm 1: 1.5 mg/m2 on days 1, 4, 8, 11 q21 days Arm 2: 1.3 mg/m2 on days 1, 4, 8, 11 + CPT 11 125 mg/m2 on day 1 q21 days | Arm 1: 1.5 mg/m2 on days 1, 4, 8, 11 q21 days Arm 2: 1.3 mg/m2 on days 1, 4, 8, 11 + gemcitabine 1000 mg/m2 on day 1 q21 days | Arm 1: 1.5 mg/m2 on days 1, 4, 8, 11 q21 days Arm 2: 1.3 mg/m2 on days 1,4,8,11 + docetaxel 75 mg/m2 on day 1 q21 |
Response rates % | NA | 10% RR | 42% RR |
Toxicity observed | Hematologic, neurotoxicity and fatigue | Abdominal pain, fatigue and thrombocytopenia | Neutropenia, neurotoxicity and fatigue |
Abbreviations: RR, response rate; CPT, irinotecan.