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. 2010 May 18;53(12):4793–4797. doi: 10.1021/jm1000248

Table 3. In Vivo Exposure Data for 1a.

dose
(mg/kg)
concentration
(μM) 0.5 h
concentration
(μM) 3 h
10 1.81 ± 0.41 0.50 ± 0.04
30 8.28 ± 0.20 3.64 ± 0.76
50 5.93 ± 1.30 6.96 ± 0.76