Figure 2.
The core molecular clock in Drosophila. CLOCK/CYCLE (CLK/CYC) bind to E-box elements (E) contained in the promoters of period ( per) and timeless (tim). PER and TIM proteins are modified by the kinases DOUBLETIME (DBT), CASEIN KINASE 2 (CK2), and SHAGGY (SGG) and the phosphatases PROTEIN PHOSPHATASE 2A (PP2A) and PROTEIN PHOSPHATASE 1 (PP1). PER and TIM dimerize and transition to the nucleus, where they repress CLK/CYC activity. Phosphorylated PER and TIM also bind the E3 ubiquitin ligase SUPERNUMERARY LIMBS (SLIMB), which leads to ubiquitination and ultimately proteolysis by the 26S proteasome.
