Table 12.
Entry | R | Substrate | Product | Yield % | ee% |
---|---|---|---|---|---|
1 | Me | 247 | 248 | 90 | 92 |
2 | Et | 248 | 249 | 86 | 94 |
3 | i-Pr | 250 | 251 | 87 | 94 |
4 | t-Bu | 252 | 253 | 86 | 94 |
5 | Ph | 254 | 255 | 87 | 88 |
6 | 4-BrPh | 256 | 257 | 78 | 85 |
7 | CH2OAc | 258 | 259 | 86 | 83 |
8 | CH2CH2OMe | 260 | 261 | 86 | 82 |
9 | CH2CH2CO2Me | 262 | 263 | 94 | 87 |