Table 4.
Chemset 8 | Aminomethyl position | % Yield | LCMS Purity |
---|---|---|---|
{2, 18} | 2 | 42 | 81 |
{3, 18} | 2 | 14 | 82 |
{1, 19} | 3 | 23 | 88 |
{2, 19} | 3 | 58 | 82 |
{3, 19} | 3 | 12 | 93 |
{1, 20} | 4 | 17 | 98 |
{2, 20} | 4 | 10 | 100 |
{3, 20} | 4 | 63 | 94 |
Chemset 8 | Aminomethyl position | % Yield | LCMS Purity |
---|---|---|---|
{2, 18} | 2 | 42 | 81 |
{3, 18} | 2 | 14 | 82 |
{1, 19} | 3 | 23 | 88 |
{2, 19} | 3 | 58 | 82 |
{3, 19} | 3 | 12 | 93 |
{1, 20} | 4 | 17 | 98 |
{2, 20} | 4 | 10 | 100 |
{3, 20} | 4 | 63 | 94 |