Table 5.
Noncompartmental pharmacokinetic parameters of DAL, HAL, and BCT
| Parameter | Analyte | ||
|---|---|---|---|
| DAL | HAL | BCT | |
| t1/2 (min) | 28.04 ± 8.55 | 16.39 ± 3.20 | 24.05 ± 4.70 |
| λz (1/min) | 0.025 ± 0.008 | 0.042 ± 0.008 | 0.029 ± 0.006 |
| AUC0-∞(μg h/L) | 579 ± 130 | 497 ± 65.8 | 595 ± 83.2 |
| CL (L/h/kg) | 2.97 ± 0.670 | 1.37 ± 0.182 | 0.183 ± 0.026 |
| AUMC (μg/L/h2) | 5063 ± 2597 | 2536 ± 800 | 4461 ± 1456 |
| MRT (h) | 0.674 ± 0.205 | 0.394 ± 0.077 | 0.578 ± 0.113 |
| Vss (L/kg) | 2.00 ± 0.030 | 0.541 ± 0.059 | 0.106 ± 0.010 |