Table 2.
Entry | Cmpd | R2 | Ar | Yield (%)a |
---|---|---|---|---|
1 | 7a | H | phenyl | 86 |
2 | 7b | H | 4-fluorophenyl | 75 |
3 | 7c | H | 3-methoxyphenyl | 62 |
4 | 7d | H | 4-methylphenyl | 68 |
5 | 7e | H | 4-methoxyphenyl | 84 |
6 | 7f | H | 4-aminophenyl | 90 |
7 | 7g | H | 3-aminophenyl | 86 |
8 | 7h | H | 2-aminophenyl | 73 |
9 | 7i | H | 3-fluorophenyl | 65 |
10 | 7j | H | 3-nitrophenyl | 97 |
11 | 7k | H | 2-methoxyphenyl | 30 |
12 | 7l | H | 2-fluorophenyl | 28 |
13 | 7m | H | 2-pyridyl | 98 |
14 | 7n | 3-Cl | phenyl | 93 |
15 | 7o | 3-methyl | phenyl | 73 |
16 | 7p | 3-CF3 | phenyl | 80 |
17 | 7q | 2,4-difluoro | phenyl | 98 |
18 | 7r | 3-pyridyl | phenyl | 94 |
Isolated yield