. 2010 Jun 9;53(13):5025–5032. doi: 10.1021/jm100456a

Table 1. The 14 Low-Micromolar TbGalE inhibitors Indentified^a.

graphic file with name jm-2010-00456a_0003.jpg

The first column shows compound structures, and the second column shows the compound identification number used throughout the text. The third column shows the IC₅₀ value of each compound as measured in enzymatic assays. The fourth and fifth columns show the EC₅₀ values as measured in whole-cell assays of T. brucei and human MRC5 cells, respectively. The final column shows the predicted LogP value of each compound.

Table 1. The 14 Low-Micromolar TbGalE inhibitors Indentifieda.

Table 1. The 14 Low-Micromolar TbGalE inhibitors Indentified^a.