Table 3.
Kinase inhibitors that directly and indirectly target Mdm2, Mdmx and p53.
| Kinase | Inhibitor |
|---|---|
| c-Abl | imatiniba [66], dasatiniba,b [67,68], nilotiniba,b [69], ON012380c [70] |
| ATM | KU-55933a [71], KU-60019a [72], CP466722 [73] |
| CDK | SNS-032 [74], AT7519a [75] |
| Chk1/Chk2 | AZD7762a [76] |
| CSN | curcumin |
| DNA-PK | morphlins [77], NU-7441a [78], NU-7422a [79], LY294002a [80]. |
| ERK | lapatiniba [81] |
| JNK | SP600125a [82] |
| MAPKAP2 | pyrazinoindolone [83], subersic acid [84], makassaric acid [84] |
| PKC | ingenol 3-angelatec [85,86], midostaurina [87], safingol [88] |
| TAF1 | apigenina [89] |
a Type I inhibitors; b Type II inhibitors; c allosteric inhibitors; d irreversible covalent inhibitors.