Table 1.
Assay | Target | Readout | Compound classes |
---|---|---|---|
Inhibitors | Purified protein | Decreased enzyme activity | ASCC |
Attenuators of denaturation | Purified protein | Increased residual enzyme activity following heat denaturation | ASCC, SCC |
Residual enzyme activity enhancers | Live cells | Increased enzyme activity in cell lysates | ASCC, SCC, alternative pathway enhancers |