. Author manuscript; available in PMC: 2010 Nov 1.

Published in final edited form as: Curr Hypertens Rev. 2009 Nov;5(4):283–306. doi: 10.2174/157340209789587717

Table 6.

Modulators of Estrogen Receptors

Agonists	Antagonists	SERMS	Phytoestrogens
Estradiol (natural) Estriol (natural) Estrone (natural) Chlorotrianisene Dienestrol Diethylstilbestrol Ethinylestradiol (ERα) Fosfestrol Mestranol Polyestradiol phosphate Quinestrol Propylpyrazole trispherol (PPT) 400x ERα Diarylpropionitrile (DPN) 30-70x ERβ	MPP (ERα) RR-tetrahydrochrysene (ERβ)	Tamoxifen 4-Hidroxytamoxifene Raloxifene Idoxifene Bazedoxifene Clomifene Toremifene Fulvestrant	Genistein (ERβ) Biochanin A (ERβ) Coumestrol Daidzein Naringenin Taxifolin Zearalenone α-zearalanol