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|
Ki (μM) |
||||
|---|---|---|---|---|
| compound | R2 | DOR | KOR | MOR |
| 1yy | 4-chloro-3- trifluoromethylphenyl | >10 | 0.10 | >10 |
| 1zz | 4-chloro-3-methylphenyl | >10 | 0.03 | >10 |
| 1aaa | 2,6-difluorophenyl | >10 | 5.00 | >10 |
| 1bbb | 2,4-dichlorophenyl | >10 | 0.29 | >10 |
