Table 1.

Yield and purity of the 1,4-disubstituted 1,2,3-triazole library members

Compd	Yield	Purity	Compd	Yield	Purity	Compd	Yield	Purity	Compd	Yield	Purity
2{1,1}	94	93	2{4,1}	92	100	2{7,1}	91	100	2{10,1}	93	81
2{1,2}	92	81	2{4,2}	94	98	2{7,2}	91	86	2{10,2}	91	100
2{1,3}	93	91	2{4,3}	93	95	2{7,3}	94	99	2{10,3}	92	84
2{1,4}	96	87	2{4,4}	92	84	2{7,4}	95	90	2{10,4}	89	84
2{1,5}	94	100	2{4,5}	92	100	2{7,5}	93	90	2{10,5}	90	100
2{1,6}	91	98	2{4,6}	96	80	2{7,6}	96	84	2{10,6}	92	82
2{1,7}	92	97	2{4,7}	96	97	2{7,7}	91	99	2{10,7}	89	94
2{1,8}	93	95	2{4,8}	90	84	2{7,8}	93	98	2{10,8}	95	83
2{1,9}	89	84	2{4,9}	92	81	2{7,9}	89	86	2{10,9}	89	100
2{2,1}	92	100	2{5,1}	94	96	2{8,1}	89	92	2{11,1}	93	86
2{2,2}	91	83	2{5,2}	91	99	2{8,2}	95	81	2{11,2}	91	96
2{2,3}	93	93	2{5,3}	95	94	2{8,3}	91	84	2{11,3}	92	86
2{2,4}	90	81	2{5,4}	92	100	2{8,4}	92	94	2{11,4}	91	86
2{2,5}	94	84	2{5,5}	94	100	2{8,5}	95	98	2{11,5}	94	98
2{2,6}	92	81	2{5,6}	93	80	2{8,6}	96	81	2{11,6}	92	81
2{2,7}	93	84	2{5,7}	92	92	2{8,7}	91	98	2{11,7}	91	100
2{2,8}	95	82	2{5,8}	90	85	2{8,8}	93	98	2{11,8}	93	95
2{2,9}	92	84	2{5,9}	92	84	2{8,9}	93	90	2{11,9}	94	95
2{3,1}	91	83	2{6,1}	92	94	2{9,1}	92	100	2{12,1}	91	81
2{3,2}	94	100	2{6,2}	96	84	2{9,2}	92	89	2{12,2}	95	97
2{3,3}	94	100	2{6,3}	91	84	2{9,3}	92	100	2{12,3}	92	93
2{3,4}	90	91	2{6,4}	93	100	2{9,4}	92	82	2{12,4}	92	81
2{3,5}	97	90	2{6,5}	93	89	2{9,5}	94	84	2{12,5}	91	98
2{3,6}	92	82	2{6,6}	95	80	2{9,6}	95	90	2{12,6}	93	84
2{3,7}	96	96	2{6,7}	93	98	2{9,7}	92	98	2{12,7}	92	96
2{3,8}	94	84	2{6,8}	93	94	2{9,8}	92	81	2{12,8}	93	84
2{3,9}	92	85	2{6,9}	89	95	2{9,9}	91	100	2{12,9}	88	82

Purities > 80% were obtained for all library members based on HPLC analysis.