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. Author manuscript; available in PMC: 2011 Dec 1.
Published in final edited form as: Biochim Biophys Acta. 2010 May 24;1806(2):183–192. doi: 10.1016/j.bbcan.2010.05.003

Table 2.

In vitro IC50 values for chemical inhibitors of PKD1

Compound IC50 (μM) Refs.
Gö6976 0.02 [119]
Gö6983 20 [119]
K252a 0.007 [119]
Staurosporine 0.04 [119]
Bisindolylmaleimide I 2 [119]
Bisindolylmaleimide II 10 [119]
Quercetin 4 [119]
Phloretin 50 [119]
Resveratrol 200 [25, 120]
CID755673 0.182 [33]
BPKDi 0.001 [34]
CRT0066101 0.001 [35]