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. Author manuscript; available in PMC: 2011 Nov 1.
Published in final edited form as: Bioorg Med Chem Lett. 2010 Aug 26;20(21):6258–6261. doi: 10.1016/j.bmcl.2010.08.096

Table 1. Ki values of 1, 2a, 2b, and 3 for rat nNOS, bovine eNOS and murine iNOS.

Kia(nM) selectivity
inhibitor
rat nNOS eNOS iNOS n/e n/i
1 7 19,000 5,800 2,700 830
2a 50 58,000 10,000 1,200 200
2b 220 59,000 13,200 270 60
3 110 58,000 21,800 530 200
a

The Ki values represent at least duplicate measurements with standard deviations of ±10%