| Analgesics |
Morphine (M6-glucuronide), pethidine (norpethidine) |
Fentanyl, levomethadone |
| Antiarrhythmic drugs |
Sotalol |
Amiodarone |
| Antibiotics |
Ciprofloxacin, levofloxacin |
Moxifloxacin |
| Antidiabetic drugs |
Glibenclamide, glimepride (hydroxy metabolite) |
Gliquidone, gliclacide |
|
Nateglinide |
Pioglitazone |
|
Sitagliptine |
|
| Anticonvulsants |
Gabapentin, pregabalin, lamotrigine, levetiracetam |
Carbamazepine, phenytoin, valproate |
| Antihypertensive drugs |
Atenolol |
Bisoprolol, carvedilol, metoprolol, propranolol |
| Cholesterol-lowering drugs |
Bezafibrate, fenofibrate |
Simvastatin, niacin |
| Drugs for gout and other rheumatological conditions |
Methotrexate |
Colchicine, hydroxychloroquine, leflunomide |
| Cardiovascular drugs |
Digoxin |
Digitoxin |
| Psychoactive drugs |
Lithium, mirtazapine |
Amitriptyline, citalopram (metabolites?), haloperidol, risperidone |
| Antiviral drugs |
Acyclovir |
Brivudine |
| Cytostatic drugs (20) |
Actinomycin D, bleomycin, capecitabine, carboplatin, cisplatin, cyclophosphamide, doxorubicin, epirubicin, etoposide, gemcitabine (dFdU), ifosfamide, irinotecan, melphalan, methotrexate, oxaliplatin, topotecan |
Anastrozole, docetaxel, doxorubicin-peg-liposomal, erlotinib, fluorouracil, gefitinib, leuprorelin, megestrol, paclitaxel, tamoxifen, terozol, vincristine, trastuzumab |