Table 2.
PAR activators and concentrations used
| PAR activator | Concentration | Selective for | Source |
|---|---|---|---|
| Thrombin | 0.01-100 nM | PAR1,3,4 | Sigma, cat T4648 |
| Cathepsin G | 1-1000 nM | PAR4 | Sigma, cat C4428 |
| Trypsin | 0.1-10 μM | PAR1,2,3,4 | Sigma, cat T9201 |
| Collagenase | 0.25% | - | Sigma, cat 4188 |
| type IV | |||
| TFLLR-NH2 | 100 μM | PAR1 | Tocris, cat 1464 |
| SFLLRN-OH (for rat) | 100 μM | PAR1 | Bachem, cat H8365 |
| SLIGRL-NH2 | 100 μM | PAR2 | Tocris, cat 1468 |
| AYPGKF-NH2 | 200 μM | PAR4 | Sigma, cat A3227 |