Table 1.
Identification of a Ligand for Palladium-Catalyzed Aerobic Allylic Acetoxylation.a
![]() | |||||
|---|---|---|---|---|---|
| Entry | Ligand | Yieldb | Entry | Ligand | Yieldb |
| 1 | None | 4% | 7 | ![]() |
0% |
| 2 |
c
|
4% | 8 | ![]() |
9% |
| 3 | ![]() |
4% | 9 | ![]() |
0% |
| 4 | ![]() |
0% | 10 | ![]() |
0% |
| 5 | ![]() |
0% | 11 | ![]() |
4% |
| 6 | ![]() |
3% | 12 | ![]() |
81% |
5% Pd(OAc)2 (3 mg, 0.0134 mmol), 5% ligand (0.0134 mmol), allyl benzene (35 μL, 0.268 mmol), AcOH (1 mL), 1 atm O2, 80 °C, 18h.
GC (internal std = nitrobenzene).
10%











