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. Author manuscript; available in PMC: 2011 Nov 1.
Published in final edited form as: Bioorg Med Chem. 2010 Sep 29;18(21):7548–7564. doi: 10.1016/j.bmc.2010.08.049

Table 3b.

Affinities (Ki=nM) of Boc-protected 3-substituted β-carbolines at αxβ3γ2(x=1–3,5,6) receptor subtypes.

Ligands α1 α2 α3 α4 α5 α6
40 graphic file with name nihms243911t27.jpg 450 5000 ND ND 5000 5000
41 graphic file with name nihms243911t28.jpg ND ND ND ND 1847 ND

ND = not determined yet (see previous tables for details of receptor binding). Data represent the average of at least three determinations with a SEM of ±5%.