Table II.
Mean Ki (nM ± SEM) |
||||
---|---|---|---|---|
A1AR | A2AAR | A2BAR | A3AR | |
ZM241385 | 3,743 ± 2,154 | 1.5 ± 1.0 | 41 ± 7 | >10,000 |
SCH58261 | 172 ± 72 | 0.8 ± 0.08 | 321 ± 57 | >10,000 |
ATL692 | 6,856 ± 2,396 | 8,809 ± 4,073 | 3.3 ± 0.8 | >10,000 |
Ki values are mean ± SEM from three or more independent experiments.