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. Author manuscript; available in PMC: 2010 Nov 22.
Published in final edited form as: J Immunol. 2009 Apr 15;182(8):4616–4623. doi: 10.4049/jimmunol.0801279

Table II.

Antagonist binding affinities for mouse adenosine receptorsa

Mean Ki (nM ± SEM)
A1AR A2AAR A2BAR A3AR
ZM241385 3,743 ± 2,154 1.5 ± 1.0 41 ± 7 >10,000
SCH58261 172 ± 72 0.8 ± 0.08 321 ± 57 >10,000
ATL692 6,856 ± 2,396 8,809 ± 4,073 3.3 ± 0.8 >10,000
a

Ki values are mean ± SEM from three or more independent experiments.