Skip to main content
. 2010 Sep 14;431(Pt 1):113–122. doi: 10.1042/BJ20100725

Table 1. Ki (app) of N-terminal reactive-site mutants for MMP-1ΔC, MMP-2, MMP-3ΔC, ADAMTS-4-2 and ADAMTS-5-4.

Ki (app) (nM)
Inhibitor MMP-1ΔC MMP-2 MMP-3ΔC ADAM17 ADAMTS-4-2 ADAMTS-5-4
N-TIMP-3 1.7±0.2 2.7±0.3 53.6±5.4 13.7±0.2 1.8±0.2 0.5±0.1
N-TIMP-3(T2G) >1000 >1000 >1000 35.6±1.9 18.3±0.1 1.5±0.1
[−1A]N-TIMP-3 800 970 >1000 33.9±2.8 22.2±0.1 1.7±0.1