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. 2010 Sep 14;431(Pt 1):113–122. doi: 10.1042/BJ20100725

Table 3. Ki (app) of position [−1] mutants for MMP-1ΔC, MMP-2, MMP-3ΔC, ADAMTS-4-2 and ADAMTS-5-4.

Ki (app) (nM)
Inhibitor MMP-1ΔC MMP-2 MMP-3ΔC ADAM17 ADAMTS-4-2 ADAMTS-5-4
[−1A]N-TIMP-3 800 970 >1000 33.9±2.8 22.2±0.1 1.7±0.1
[−xG]N-TIMP-3 >1000 >1000 >1000 465 107 118
[−ME]N-TIMP-3 >1000 >1000 >1000 529 326 327
[−MM]N-TIMP-3 >1000 >1000 >1000 153 75.7 69.4
[−MK]N-TIMP-3 500 750 >1000 325 280 217