TABLE 2.
Plasma protein binding of VU591
Percentage VU591, warfarin (control), and verapamil (control) bound to human or rat serum protein are shown. Data are mean ± S.D. from 2 replicate experiments.
| Human | Rat | |
|---|---|---|
| % bound | ||
| VU591 | 99.14 ± 0.0056 | 98.39 ± 0.0010 |
| Warfarin | 99.62 ± 0.0002 | 99.57 ± 0.0003 |
| Verapamil | 93.41 ± 0.0088 | 97.14 ± 0.0037 |