Table 4A.
Parameters (units) | CMAB009 dose (mg/m2) | ||
100 | 250 | 400 | |
Ke (h−1) | 0.015 ± 0.002 | 0.009 ± 0.001 | 0.009 ± 0.002 |
Tl/2ke (h) | 47.47 ± 6.61 | 78.42 ± 6.23 | 83.58 ± 15.86 |
AUC0-t (µg.h/mL) | 2939.01 ± 569.47 | 15525.30 ± 4797.02 | 26615.95 ± 4827.53 |
AUCt-∞ (µg.h/mL) | 16.59 ± 11.46 | 39.51 ± 23.46 | 1561.42 ± 1294.44 |
AUC0-∞ (µg.h/mL) | 2955.60 ± 571.57 | 15564.81 ± 4812.12 | 28177.37 ± 5647.10 |
AUC0-t % | 99.43 ± 0.35 | 99.76 ± 0.10 | 94.80 ± 3.77 |
MRT (h) | 66.66 ± 3.98 | 124.43 ± 20.90 | 121.79 ± 22.24 |
C//F (mL/h.m2) | 34.81 ± 7.55 | 17.63 ± 6.18 | 14.68 ± 2.93 |
VSS (mL/m2) | 2300.28 ± 348.73 | 2116.88 ± 526.31 | 1745.34 ± 258.95 |