Table 2.
Entry | R' | R | Yielda (%) |
1 | H | H | 95 |
2 | H | 4-OH | 93 |
3 | 2'-OH | H | 91 |
4 | H | 3,4-O-CH2-O- | 90 |
5 | 4'-OH | 4-OH | 94 |
6 | 4'-OMe | 4-Cl | 88 |
7 | 4'-OH | 4-OMe | 82 |
8 | H | 4-NO2 | 82 |
9 | H | 3,4-OH | 87 |
10 | 2'-OH | 3-OMe, 4-OH | 81 |
11 | 3'-OH | 2-NO2 | 81 |
12 | 4'-OMe | 4-OMe | 79 |
13 | 4'-OH | 3,4-OH | 86 |
14 | 4'-OCH2CH = CH2 | 4-OMe | 85 |
15 | 2',4'-OMe | 4-OMe | 89 |
a Isolated pure yield.