Table 1.
Drug Activities Across Leukemia and CNS Cell Lines and Summary Statistics for Complete NCI-60 Cell Line Screen
| NSC number | FdUMP(10) | Fluorouracil (5FU) | Floxuridine (FUdR) | Topotecan HCl | Irinotecan HCl |
|---|---|---|---|---|---|
| 697912 | 19893 | 27640 | 609699 | 616348 | |
| CNS:SF-268 | 8.30 | 4.30 | 6.53 | 7.92 | 5.41 |
| CNS:SF-295 | 8.30 | 4.30 | 6.50 | 7.69 | 5.14 |
| CNS:SF-539 | 8.30 | 5.88 | 6.53 | 7.89 | 5.30 |
| CNS:SNB19 | 6.77 | 3.94 | 5.91 | 7.66 | 4.62 |
| CNS:SNB75 | 6.45 | 3.74 | 6.03 | 7.68 | 4.80 |
| CNS:U251 | 6.94 | 4.35 | 6.35 | 7.79 | 5.39 |
| LE:CCRF-CEM | na | 4.48 | 6.41 | 8.07 | 5.46 |
| LE:HL-60 | 7.90 | 4.68 | 6.27 | 7.85 | 4.95 |
| LE:K-562 | 5.63 | 4.68 | 6.11 | 7.22 | 4.96 |
| LE:MOLT-4 | 8.28 | 4.87 | 6.44 | 8.06 | 5.78 |
| LE:RPMI-8226 | 6.64 | 5.31 | 5.74 | 6.61 | 4.69 |
| LE:SR | 8.30 | 5.38 | 6.50 | 7.66 | 6.63 |
| NCI-60 Minimum | 4.30 | 3.31 | 3.61 | 5.45 | 4.08 |
| NCI-60 Maximum | 8.30 | 5.98 | 6.58 | 8.07 | 6.63 |
| NCI-60 Average | 7.15 | 4.64 | 5.83 | 7.19 | 4.89 |
| NCI-60 Range | 4.00 | 2.67 | 2.96 | 2.63 | 2.55 |
Drug activities are GI50’s, presented as −log10 values.
Drug activities obtained from http://dtp.nci.nih.gov/dtpstandard/cancerscreeningdata/index.jsp.