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. 2010 Oct 26;2011:727241. doi: 10.1155/2011/727241

Table 1.

Examples of therapeutic applications using monocyte/macrophage-targeted liposomes.

Ligand Active Disease Reference
Anionic lipids
Dexamethasone Atherosclerosis [22]
SLPI Inflammatory lung disease [23]
Bisphosphonates Restnosis [24]
Rifampicin Tuberculosis [25]
Dideoxycytidine-5′-triphosphate HIV [26]
Clarithromycin Mycobacterium avium infection [27]

Peptides
Muramyl tripeptide (MTP) MTP-phosphotidylethanolamine Osteosarcoma [28]
Arg-Gly-Asp (RGD) Diclofenac sodium (model drug) Cerebrovascular disease [29]

Antibodies
Anti-VCAM-1 Prostaglandins Atherosclerosis [30]
Anti-CC52 Colon Cancer [31]
Anti-CC531 Colon Adenocarcinoma [32]
Anti-CD11c/DEC-205 tumour antigen (OVA) Cancer [21]

Lectins
Mann-C4-Chol Dexamethasone palmitate Inflammatory lung disease [33]
Man2DOG [34]
Aminophenyl-α-D-mannopyranoside Doxorubicin Experimental visceral leishmaniasis [6]
Ciprofloxacin Respiratory infection [5]
Man3-DPPE OVA [35]
Gastric cancer [36]

Other Ligands
Maleylated bovine serum albumin (MBSA) [25]
O-steroly amylopectin (O-SAP) [25]
Fibronectin [37]
Galactosyl [37]