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. Author manuscript; available in PMC: 2012 Apr 14.
Published in final edited form as: J Med Chem. 2011 Mar 4;54(7):2409–2421. doi: 10.1021/jm101549k

Table 5.

Plasma PK profile of 7 (1 mg/kg i.v. & 1 mg/kg p.o.) in Sprague-Dawley rats administered in PBS

Route AUC last (ng · h/mL) AUC/Dose (ng · h/mL/dose) T1/2 (h) Cl (mL/min/kg) Vss (L/kg) Cmax (ng/mL) Tmax (h) F (%)
i.v. 121 126 0.95 133 9.0 - - -
p.o. 124 124 1.4 - - 55 0.75 98
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