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. Author manuscript; available in PMC: 2012 Mar 15.
Published in final edited form as: Acc Chem Res. 2010 Dec 22;44(3):180–193. doi: 10.1021/ar1001186

Figure 1.

Figure 1

(A) Typical Aspartic Acid Protease Active Site, (B) Comparison of Amide. and Pyrrolinone Units, (C) Design of 3,5- and 2,5-Pyrrolinones, (D) Registrations of 3,5- and 2,5-Linked Pyrrolinone Scaffolds.