Table 6.
Intracellular diamidine concentration after 1 h of exposure to 10 μM permeant
Cell line | Source condition | Diamidine concn (μM ± SEM) |
||
---|---|---|---|---|
DB75 | DB820 | CPD0801 | ||
s427 | Ex vivo | 596 ± 203 | 264 ± 22 | 64.0 ± 13 |
In vitro | 12.6 ± 2.2 | 0.43 ± 0.12 | 0.15 ± 0.03 | |
tbat1−/− | Ex vivo | 21.3 ± 1.7 | 5.70 ± 0.22 | 1.12 ± 0.42 |
In vitro | 12.2 ± 4.0 | 0.24 ± 0.05 | 0.15 ± 0.03 |