Table 1.
Compound and cell line | EC50 (nM) | CC50 (μM) | Selective indexa |
---|---|---|---|
4′-C-Me-2′-dA | |||
HOS | 63 ± 7 | 59 ± 5 | 936 |
TZM-bl | 69 ± 4 | 169 ± 22 | 2,550 |
4′-C-Et-2′-dA | |||
HOS | 221 ± 3 | 369 ± 22 | 1,669 |
TZM-bl | 184 ± 20 | 204 ± 28 | 1,109 |
Selective index = CC50/EC50.